CB 1 receptor

Cannabinoid CB1 receptor antagonism modulates plasma corticosterone in rodents

Therapeutic drug monitoring / Mice / Animals / Corticosterone / Male / Rats / Time Dependent / Time Factors / Reproducibility of Results / Wistar Rats / Biological markers / Pyrazoles / Knockout Mice / CB 1 receptor / Piperidines / Rats / Time Dependent / Time Factors / Reproducibility of Results / Wistar Rats / Biological markers / Pyrazoles / Knockout Mice / CB 1 receptor / Piperidines

PAPEL DE LOS ENDOCANABINOIDES EN ATEROSCLEROSIS: RELACIÓN CON LA FUNCIÓN ENDOTELIAL

Cardiovascular Risk / Metabolic syndrome / Nitric oxide / Endothelial Function / CB 1 receptor

Diaryl piperidines as CB1 receptor antagonists

Organic Chemistry / Obesity / Diet / Mice / Animals / Eating / Food intake / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / CB 1 receptor / Piperidines / Eating / Food intake / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / CB 1 receptor / Piperidines

Cannabinoides endógenos en la enfermedad hepática: muchos dardos para una sola diana

Gastroenterology / Obesity / Inflammation / Apoptosis / Energy Metabolism / Liver diseases / Humans / Portal hypertension / Liver Cirrhosis / Fatty acids / Mice / Blood Pressure / Animals / Liver Fibrosis / Hepatic Stellate Cells / Clinical Sciences / Rats / Monocytes / Liver Disease / Neurosciences / Ascites / CB 1 receptor / Arachidonic Acid / Vascular Resistance / Liver diseases / Humans / Portal hypertension / Liver Cirrhosis / Fatty acids / Mice / Blood Pressure / Animals / Liver Fibrosis / Hepatic Stellate Cells / Clinical Sciences / Rats / Monocytes / Liver Disease / Neurosciences / Ascites / CB 1 receptor / Arachidonic Acid / Vascular Resistance

Diaryl piperidines as CB1 receptor antagonists

Organic Chemistry / Obesity / Diet / Mice / Animals / Eating / Food intake / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / CB 1 receptor / Piperidines / Eating / Food intake / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / CB 1 receptor / Piperidines

Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide (SR141716) a potent CB1 receptor antagonist

Organic Chemistry / Pharmaceutical Chemistry / Mice / Animals / Drug Design / Molecular Conformation / Bioorganic and medicinal Chemistry / Pyrazoles / CB 1 receptor / Piperidines / Molecular Conformation / Bioorganic and medicinal Chemistry / Pyrazoles / CB 1 receptor / Piperidines

Cannabinoides endógenos en la enfermedad hepática: muchos dardos para una sola diana

Gastroenterology / Obesity / Inflammation / Apoptosis / Energy Metabolism / Liver diseases / Humans / Portal hypertension / Liver Cirrhosis / Fatty acids / Mice / Blood Pressure / Animals / Liver Fibrosis / Hepatic Stellate Cells / Clinical Sciences / Rats / Monocytes / Liver Disease / Neurosciences / Ascites / CB 1 receptor / Arachidonic Acid / Vascular Resistance / Liver diseases / Humans / Portal hypertension / Liver Cirrhosis / Fatty acids / Mice / Blood Pressure / Animals / Liver Fibrosis / Hepatic Stellate Cells / Clinical Sciences / Rats / Monocytes / Liver Disease / Neurosciences / Ascites / CB 1 receptor / Arachidonic Acid / Vascular Resistance

Cannabinoides endógenos en la enfermedad hepática: muchos dardos para una sola diana

Gastroenterology / Obesity / Inflammation / Apoptosis / Energy Metabolism / Liver diseases / Humans / Portal hypertension / Liver Cirrhosis / Fatty acids / Mice / Blood Pressure / Animals / Liver Fibrosis / Hepatic Stellate Cells / Clinical Sciences / Rats / Monocytes / Liver Disease / Neurosciences / Ascites / CB 1 receptor / Arachidonic Acid / Vascular Resistance / Liver diseases / Humans / Portal hypertension / Liver Cirrhosis / Fatty acids / Mice / Blood Pressure / Animals / Liver Fibrosis / Hepatic Stellate Cells / Clinical Sciences / Rats / Monocytes / Liver Disease / Neurosciences / Ascites / CB 1 receptor / Arachidonic Acid / Vascular Resistance
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